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      1. 原料藥及中間體服務

        吉林天衡原料藥和中間體生產基地位于河南省鄧州市工業園區南陽天衡制藥廠,車間占地1萬平米,各類型反應釜40余臺。依托北京天衡藥物研究院有限公司產品的研發 ,已完成小試品種有100多個,目前工業化規模生產13個品種,產品質量達到國際高水平。產品出口日本、印度、東南亞和歐洲部分國家。


        原料藥及中間體服務產品目錄



        產品名稱Product nameCAS登記號(CAS No.)標準Specification結構式Structural Formula
        伏格列波糖及中間體
        Voglibose & Intermediates
        伏格列波糖
        Voglibose
        83480-29-9JP16
        IP
        In house
         01
        2,3,4,6-四-O-芐基-α-D-葡萄糖
        2,3,4,6-Tetra-O-benzyl-α-D-glucopyranose
        4132-28-9
        6564-72-3
        ≥99%
        In house
         02
        (2R,3S,4S,5S)-5-羥基-2,3,4-三 (芐氧基)-5-[(芐氧基)甲基]-環己酮 (2R,3S,4S,5S)-5-Hydroxy-2,3,4-tris (phenylmethoxy)-5-[(phenylmethoxy)methyl]-cyclohexanone115250-38-9≥99%
        In house
         03
        四芐基伏格列波糖
        Tetra-Benzyl-Voglibose
        115250-39-0≥99%
        In house
         04
        鹽酸吉西他濱中間體Gemcitabine Hydrochloride Intermediate2-脫氧-2,2二氟-戊呋喃糖-1-酮- 3,5-二苯甲酸酯(T6) 2-Deoxy-2,2-difluoro-D-erythro-pentafuranous-1-ulose-3,5-dibenzoate122111-01-7≥99%
        In house
         05
        帕利哌酮及中間體
        Paliperidone & Intermediates
        帕利哌酮
        Paliperidone
        144598-75-4≥99%
        In house
         06
        帕利哌酮棕櫚酸酯
        Paliperidone Palmitate
        199739-10-1≥99%
        In house
         07
        3-(2-氯乙基)-6,7,8,9-四氫-9-羥基-2-甲基-4H-吡啶并[1,2-a]嘧啶-4-酮3-(2-Chloroethyl)-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one130049-82-0≥99%
        In house
         08
        6-氟-3-哌啶-4-基-1,2-苯并異噁唑鹽酸鹽
        6-Fluoro-3-(4-piperidinyl)-1,2-
        benzisoxazole hydrochloride
        84163-13-3≥99%
        In house
         09
        鹽酸厄洛替尼中間體
        Erlotinib Hydrochloride
        Intermediates
        6,7-雙(甲氧基乙氧基)喹唑啉酮
        6,7-Bis-(2-methoxyethoxy)-4(3H)-quinazolinone
        179688-29-0≥99%
        In house
         10
        阿加曲班及中間體Argatroban &
        Intermediate
        阿加曲班
        Argatroban Hydrate
        74863-84-6≥99%
        In house
         11
        (2R,4R)-4-甲基-2-哌啶甲酸乙酯
        Ethyl (2R,4R)-4-methyl-2-piperidinecarboxylate
        74892-82-3≥99%
             In house
         12
        帕布昔利布及中間體Palbociclib & Intermediates帕布昔利布(帕博西尼)
        Palbociclib
        571190-30-2≥99%
        In house
         13
        4-(6-氨基吡啶-3-基)哌嗪-1-羧酸叔丁酯
        4-(6-Aminopyridin-3-yl)piperazine-1-carboxylic acid tert-butyl este
        571188-59-5≥99%
        In house
         14
        6-溴-2-氯-8-環戊基-5-甲基-吡啶并[2,3-D]嘧啶-7(8H)-酮6-bromo-2-chloro-8-cyclopentyl-5-Methylpyrido[2,3-d]pyriMidin-7(8H)-one1016636-76-2≥99%
        In house
         15
        奧格列汀Omarigliptin & IntermediatesN-[(2R,3S)-2-(2,5-二氟苯基)四氫-5-氧代-2H-吡喃-3-基]氨基甲酸叔丁酯N-[(2R,3S)-2-(2,5-Difluorophenyl)tetrahydro-5-oxo-2H-pyran-3-yl]carbamic acid 1,1-dimethylethyl ester951127-25-6≥99%
        In house
         16
        2-(甲基磺?;?-2,4,5,6-四氫吡咯并[3,4-c]吡唑苯磺酸鹽
        2,4,5,6-Tetrahydro-2-(methylsulfonyl)pyrrolo[3,4-c]pyrazole benzenesulfonate
        1280210-80-1≥99%
        In house
         17


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